jinxianda biotechnology
Dinotefuran, an organic substance, is used primarily as an insecticide.
Product chemical information:
Product name: Dinotefuran
International common name: Dinotefuran,
CAS No.: 16525270-0
CPAC No.: 749
Chemical name: dinotefuran (bsi,pa iso); mti-446; DINOTEFURAN STANDARD; 1-Methyl-2-nitro-3-(tetrahydro-3-furylmethyl)guanidine; 2-methyl-1-nitro-3-(tetrahydrofuran-3-ylmethyl)guanidine; 2-methyl-1-nitro-3-(tetrahydrofuran-2-ylmethyl)guanidine
Structural formula:
Category: Pesticides
Molecular formula: C7H14N4O3
Relative molecular weight: 202.2
Physical and chemical properties:
Melting point: 107.5℃:
Boiling point: 208℃ decomposition
Vapor pressure (30℃): <1.7×103mPa;
Octanol/water partition coefficient: KowlogP=-0.549(25℃);
Density: 140:
Henry's constant: 8.7×10-9Pam3mo。
Solubility (g/L,25℃): Water 39.8: Hexane 9.0×10-6, heptane 11×10-6, xylene 72×10-3, toluene 150×10-3, dichloromethane 11, acetone 58, methanol 57, ethanol 19, ethyl acetate 5.2. Stability: Stable at 150℃, hydrolyzed DTS > for 1 year (pH4.0, pH7.0 and pH9.0); The photolysis DT50 in water was 3.8h
Product characteristics
Advantages: the only nicotinic insecticide containing tetrahydrofuran ring has excellent control effect on the puncture and suction mouth pests. It not only has the activities of tentacling, gastric toxicity and root inhalation, but also has the characteristics of strong endosperm, low dosage, good quick effect, high activity, long lasting effect, wide insecticidal spectrum and so on
Main crops and control targets: In rice, wheat, vegetables, fruit trees, tea, cotton, tobacco and other crops, mainly used for the prevention and control of various plant hopper, bugs, mealworms, leafhoppers, leaf flies, thrips, jump, aphids and leaf moth, small peach budworm, rice borers, plutella xylostella, caterpillar, etc., and the white mosquitoes, cockroaches, fleas, housefly, mosquitoes and other health pests.
Patent Overview
Compound patents at home and abroad
(1)Domestic compound patent
Patent number: CN1099418C;
Patent name: (tetrahydro3-furanyl) methylamine;
Application date: 1994-10-26
The patentee: Mitsui Chemical Co
(2)Patent of foreign compounds
Patent number: EP649845A1;
Patent name: Furanyl insecticide;
Application date: 1994-10-26:
The patentee: Mitsui Toatsu Chemicals InC
Domestic and overseas market overview
Overseas market: The average annual growth rate for the five years from 2004 to 2009 was 20.8%. In 2005, the product entered South Korea and the United States, and in 2008, it was listed in the European Union. The average annual value of dinotefuran in the Japanese market reached 110 million USD in 2011 and 2012.
Domestic market: This product is not used for a long time in China, is currently under the "crazy" registration period. At home, its use area will gradually expand, the future will appear the market competition is white hot! In 2016, Hubei Plant Protection Station will focus on promoting pesticide and medical device varieties.
International agrochemical company in the foreign registration of excellent product formula recommendation
Country | Active ingredients and content | Dosage form | Control object | Registered company |
U.S. | 0.96%, 20.0% Dinotefuran | soluble concentrate | Moths, thrips, borers, sticky worms and other pests | Mitsui chemicals agro, inc. |
20.0% Dinotefuran | missible oil | It is used to control mosquito, ant, moth and crickets on ornamental plants, houses and building materials. | ||
0.50% Dinotefuran | granules | Cockroaches, houseflies | Valent biosciences corporation |
|
70.0% Dinotefuran | missible oil | Used to control leafminer flies, beetles, whitefly, aphids, etc. on fruits and vegetables | Valent u.s. a. corporation |
|
Japan | 0.01% Dinotefuran | fluid | Bemisia tabaci, aphids, thrips, melon leaf nail, mealworms, stink bug, beetles and other pests on pepper, eggplant, tomato and other cigars, melons and squash, radishes and cabbage and other cruciferous leaf vegetables, peas and other beans and purple sunflower | MITSUI CHEMICALS |
0.3% ethofenprox +0.5% Dinotefuran |
powder | Rice planthopper, stink bug, locust, rice borers | ||
0.01% Dinotefuran +0.01% penthiopyrad |
wettable powder | Eggplant, tomato, cherry tomato, green pepper, cucumber, Chinese cabbage, lettuce, lettuce, green onion, rose (ornamental flowers, plants) powdery mildew, leaf mildew, scab, aphids, mealworms, thrips, aphids, leaf wasp, etc | ||
1% Dinotefuran +4% benfuracarb |
granules | Leaf roller, rice water weevils | OATアグリオ Co., Ltd. | |
4% metominostrobin +1.67% Dinotefuran |
granules | Rice blast, ear blight, smut, rice black tail leafhopper, planthopper, stink bug, etc | Beixing Chemical Industry Co., Ltd. | |
4% Dinotefuran +48% probenazole |
wettable powder | Rice planthopper, rice water weevil, rice blast disease | ||
12% rabicide +5% Dinotefuran |
wettable powder | Rice blast, lychee bug, rice planthopper, black - tailed leafhopper | ||
5% Dinotefuran +20% thiophanate-methyl |
wettable powder | Rice blast, sheath blight, smut, rice planthopper, stink bug, black tail leafhopper and other diseases and insect pests | Beixing Chemical Co., Ltd. | |
4% Chlorantraniliprole +15% Dinotefuran |
wettable powder | Insect insects such as aphids, rapeseed beetles, twill moth, diamondback moth, thrips, borers, sticky worms and so on | Mitsui Chemical Agro Co. Ltd | |
7% ethofenprox +3% dinotefuran | wettable powder | Rice planthopper, rice thrips, black tailed leafhoppers, rice leaf roller, stink bug | ||
9% Dinotefuran+18% buprofezin | wettable powder | Rice planthoppers, black-tailed leafhoppers, stink bugs | Japan Pesticide Corporation |
The first registration information of domestic active drugs and preparations and the current pneumatic product registration situation analysis
Active drug (master drug) | |||||
The registration number | Active ingredients | Content | Dosage form | Control object | Production enterprise |
PD2016353 | Dinotefuran | 99.10% | Active drug | - | Mitsui Chemical Agro Co. Ltd |
Single preparation | |||||
The registration number | Active ingredients | Content | Dosage form | Control object | Production enterprise |
PD20160354 | Dinotefuran | 20% | Soluble granule | Rice borer, planthopper, cucumber (protected area) thrips, white whitefly | Mitsui Chemical Agro Co. Ltd |
Active ingredients | Content | Dosage form | Crops | Prevention objects |
Dinotefuran·ethofenprox | 9%+18% | suspending agent | paddy | plant hopper |
Dinotefuran·imidacloprid | 5%+30% | suspending agent | cowpeas | thrips |
Dinotefuran·buprofezin | 5%+25% | suspending agent | Citrus trees | Scale insect |
Dinotefuran·isoprocarb | 4%+20% | suspending agent | paddy | Rice planthopper |
Dinotefuran·indoxacarb | 10%+10% | suspending agent | Peach trees | peach fruit moth |
Dinotefuran·pyridyne | 5%+10% | suspending agent | Citrus trees | Scale insects |
Dinotefuran·dimehypo | 0.1%+0.3% | granules | paddy | Chilo suppressalis/Rice planthopper |
Dinotefuran·pyridaben | 40%+20% | water dispersible granule | cabbage | Phyllotreta vittata Fabricius |
Dinotefuran·thiamethoxam | 5%+15% | water dispersible granule | paddy | Rice planthopper |
Dinotefuran·pymetrozine | 10%+40% | water dispersible granule | paddy | Rice planthopper |
Dinotefuran·monosultap | 20%+60% | water dispersible granule | paddy | Chilo suppressalis/Rice planthopper |
Dinotefuran·fludioxonil | 7.5%+2.5% | seed treatmentsuspending agent | paddy | Bakanae disease/plant hopper |
Dinotefuran·tebuconazole | 14.7%+0.3% | seed treatmentsuspending agent | wheat | Scatter smut/aphid |
Dinotefuran·bifenthrin | 0.4%+0.5% | granules | cabbage | Phyllotreta vittata Fabricius |
Dinotefuran·spirotetramat | 10%+10% | suspending agent | Citrus trees | Scale insects |
Dinotefuran·Tolfenpyrad | 24%+40% | water dispersible granule | paddy | thrips |
Dinotefuran·nitenpyram | 15%+45% | water dispersible granule | paddy | Rice planthopper |
Dinotefuran·Thifluzamide | 7.5%+7.5% | seed treatmen tdispersible powder | wheat | Sheath blight/aphids |
Dinotefuran·flonicamid | 10%+2% | Dispersible oil suspending agent | cucumber | aphids |
Dinotefuran·Beta-cyhalothrin | 16%+8% | water dispersible granule | cucumber | whitefly |
Product packaging
Product label